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Search Results for " Cholecystokinin Receptor "

ターゲット

35

阻害剤

1

リコンビナントタンパク質

カタログ番号 製品名 別名 ターゲット
TP1197 Sincalide SQ19844,CCK-8,Cholecystokinin octapeptide Others
Sincalide (CCK-8) is a cholecystokinetic drug administered by injection to aid in diagnosing disorders of the gallbladder and pancreas. It is the 8-amino acid C-terminal fragment of cholecystokinin.
TQ0062 Nastorazepide Z-360 cholecystokinin
Nastorazepide (Z-360) is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic activity.
T2312 Loxiglumide CR-1505 cholecystokinin
Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.
T4579 Pentagastrin ICI-50123 Others , cholecystokinin
Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis of salivary proteins.
T14932 Ceruletide Cerulein,Caerulein,FI-6934 cholecystokinin
Ceruletide (Caerulein) is a potent agonist of cholecystokinin receptor and it also is a safe and effective cholecystokinetic agent. It has a direct spasmogenic effect on the gallbladder muscle and bile ducts.
T1052 Proglumide cholecystokinin
Proglumide (Binoside) is a cholecystokinin antagonist, which blocks both the CCKA and CCKB subtypes. Proglumide is a drug that exerts an inhibitory effect on gastric secretion and reduces gastrointestinal motility. It is...
T27503 GV150013 GV 150013,GV-150013 cholecystokinin
GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
T34123 Pranazepide FR120480,FK 480,FR-120480 cholecystokinin
Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders and pancreatitis.
T15382 GI 181771 cholecystokinin
GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity.
T14932L1 Ceruletide Ammonium Salt Caerulein Ammonium Salt,Ceruletide Ammonium Salt(17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt cholecystokinin
Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is a potent cholecystokinin receptor agonist and a safe and effective cholecystokinin receptor agonist with direct spasmodic e...
TP2030L1 Gastrin I (human) acetate Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate cholecystokinin
Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (CCK2) receptor.
T9343 N-Cbz-DL-tryptophan cholecystokinin
N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.
T12404 CCK-A receptor inhibitor 1 cholecystokinin
T14932L Ceruletide Ammonium acetate FI-6934 Ammonium acetate,Caerulein Ammonium acetate,Ceruletide Ammonium acetate (17650-98-5 free base) cholecystokinin
Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist. Ceruletide Ammonium acetate is a safe and effective cholecystokinetic agent and small bowel and exocrine pancreatic stim...
T26971 Ceclazepide
Ceclazepide is an antagonist of cholecystokinin receptor.
T26483 A-65186 A65186
A 65186 is a Type A Cholecystokinin (CCK) receptor antagonist.
T24202 Jmv 167 Jmv-167,Jmv167
Jmv 167 is an antagonist of the Cholecystokinin receptor.
T23886 Cholecystokinin (27-32)-amide Cholecystokinin (27-32)-NH2
Cholecystokinin (27-32)-amide is a CCK receptor antagonist.
T29502 A 70874 A-70874,A70874
A70874 has high selectivity and potency for cholecystokinin (CCK) a receptor.
T28613 RP73870 RP 73870,RP-73870
RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.
T25552 Jmv 320 Jmv-320,Jmv320
Jmv 320 is a highly selective gastrin receptor and cholecystokinin receptor antagonist. It is a cyclic cholecystokinin-8 analog in which positions 28 and 31 have been replaced by Lys, with their side chains bridged by a ...
T22895 L-365260 L-365,260 Others
cholecystokinin receptor 2 (CCK2) antagonist
T13261 CCK-B Receptor Antagonist 1 Others
CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
T24204 Jmv 179 Jmv-179,Jmv179
Jmv 179 is an antagonist of the cholecystokinin receptor.
T24293 L 368935 L-368935,L368,935,L-368,935,L 368,935,L368935
L 368935 is an antagonist of the cholecystokinin receptor.
T27664 JNJ-17156516 JNJ17156516,JNJ 17156516
JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.
T28335 PD 140376 PD-140376,PD140376
PD 140376 is a highly selective antagonist radioligand for the cholecystokinin(B)-gastrin receptor in guinea pig gastric mucosa & cerebral cortex in the peripheral and central nervous systems.
T27669 JNJ-26070109 JNJ26070109
JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.
T28331 PD 136450 Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189
Cholecystokinin type B receptor antagonist PD-136,450 is a partial secretory agonist in the stomach and a full agonist in the pancreas of the rat. Gastrin (cholecystokinin type B (CCK-B)) receptor antagonists may help to...
T68482 CE-326597
CE-326597 is a potent and selective CCK1R agonist. The type 1 cholecystokinin receptor (CCK1R) has multiple physiologic roles relating to nutrient homeostasis,including mediation of postcibal satiety. The type 1 cholecy...
T15101 Devazepide L-364,718,MK-329 Others
Devazepide is a competitive and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor (IC50s: 81 pM, 45 pM, and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respective...
T17274 YM022 CCR
YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki v...
T28612 RP-72540 RPR 102681,RPR-102681,RPR102681
RP-72540 is a cholecystokinin B receptor antagonist. RP 72540 showed selectivity factors in express of 200 for CCKA versus CCKB receptors and also had high affinity for gastrin binding sites in the stomach. Administratio...
T62039 L-365260 hemihydrate
L-365260 hemihydrate is a selective, orally active non-peptide gastrin and brain cholecystokinin receptor (CCK-B) antagonist, demonstrating competitive interaction with guinea pig stomach gastrin and brain CCK receptors ...
T8761 [Leu15]-Gastrin I human Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2 Others
[Leu15]-Gastrin I human (Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2) encodes for the protein [Leu15]-Gastrin I in human. In human chromosome, the gene GAST is localized on...

Compounds

Sincalide
TP1197
Synonym: SQ19844,CCK-8,Cholecystokinin octapeptide
Target: Others
Nastorazepide
TQ0062
Synonym: Z-360
Target: cholecystokinin
Loxiglumide
T2312
Synonym: CR-1505
Target: cholecystokinin
Pentagastrin
T4579
Synonym: ICI-50123
Target: Others, cholecystokinin
Ceruletide
T14932
Synonym: Cerulein,Caerulein,FI-6934
Target: cholecystokinin
Proglumide
T1052
Synonym:
Target: cholecystokinin
GV150013
T27503
Synonym: GV 150013,GV-150013
Target: cholecystokinin
Pranazepide
T34123
Synonym: FR120480,FK 480,FR-120480
Target: cholecystokinin
GI 181771
T15382
Synonym:
Target: cholecystokinin
Ceruletide Ammonium Salt
T14932L1
Synonym: Caerulein Ammonium Salt,Ceruletide Ammonium Salt(17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt
Target: cholecystokinin
Gastrin I (human) acetate
TP2030L1
Synonym: Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate
Target: cholecystokinin
N-Cbz-DL-tryptophan
T9343
Synonym:
Target: cholecystokinin
CCK-A receptor inhibitor 1
T12404
Synonym:
Target: cholecystokinin
Ceruletide Ammonium acetate
T14932L
Synonym: FI-6934 Ammonium acetate,Caerulein Ammonium acetate,Ceruletide Ammonium acetate (17650-98-5 free base)
Target: cholecystokinin
Ceclazepide
T26971
Synonym:
Target:
A-65186
T26483
Synonym: A65186
Target:
Jmv 167
T24202
Synonym: Jmv-167,Jmv167
Target:
Cholecystokinin (27-32)-amide
T23886
Synonym: Cholecystokinin (27-32)-NH2
Target:
A 70874
T29502
Synonym: A-70874,A70874
Target:
RP73870
T28613
Synonym: RP 73870,RP-73870
Target:
Jmv 320
T25552
Synonym: Jmv-320,Jmv320
Target:
L-365260
T22895
Synonym: L-365,260
Target: Others
CCK-B Receptor Antagonist 1
T13261
Synonym:
Target: Others
Jmv 179
T24204
Synonym: Jmv-179,Jmv179
Target:
L 368935
T24293
Synonym: L-368935,L368,935,L-368,935,L 368,935,L368935
Target:
JNJ-17156516
T27664
Synonym: JNJ17156516,JNJ 17156516
Target:
PD 140376
T28335
Synonym: PD-140376,PD140376
Target:
JNJ-26070109
T27669
Synonym: JNJ26070109
Target:
PD 136450
T28331
Synonym: Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189
Target:
CE-326597
T68482
Synonym:
Target:
Devazepide
T15101
Synonym: L-364,718,MK-329
Target: Others
YM022
T17274
Synonym:
Target: CCR
RP-72540
T28612
Synonym: RPR 102681,RPR-102681,RPR102681
Target:
L-365260 hemihydrate
T62039
Synonym:
Target:
[Leu15]-Gastrin I human
T8761
Synonym: Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2
Target: Others

Recombinant Proteins

カタログ番号 製品名 Species Expression System
TMPH-03099 Aminopeptidase N/CD13 Protein, Pig, Recombinant (His & Myc) Sus scrofa (Pig) E. coli
Broad specificity aminopeptidase which plays a role in the final digestion of peptides generated from hydrolysis of proteins by gastric and pancreatic proteases. Also involved in the processing of various peptides includ...