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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TP1197 | Sincalide | SQ19844,CCK-8,Cholecystokinin octapeptide | Others |
Sincalide (CCK-8) is a cholecystokinetic drug administered by injection to aid in diagnosing disorders of the gallbladder and pancreas. It is the 8-amino acid C-terminal fragment of cholecystokinin. | |||
TQ0062 | Nastorazepide | Z-360 | cholecystokinin |
Nastorazepide (Z-360) is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic activity. | |||
T2312 | Loxiglumide | CR-1505 | cholecystokinin |
Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor. | |||
T4579 | Pentagastrin | ICI-50123 | Others , cholecystokinin |
Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis of salivary proteins. | |||
T14932 | Ceruletide | Cerulein,Caerulein,FI-6934 | cholecystokinin |
Ceruletide (Caerulein) is a potent agonist of cholecystokinin receptor and it also is a safe and effective cholecystokinetic agent. It has a direct spasmogenic effect on the gallbladder muscle and bile ducts. | |||
T1052 | Proglumide | cholecystokinin | |
Proglumide (Binoside) is a cholecystokinin antagonist, which blocks both the CCKA and CCKB subtypes. Proglumide is a drug that exerts an inhibitory effect on gastric secretion and reduces gastrointestinal motility. It is... | |||
T27503 | GV150013 | GV 150013,GV-150013 | cholecystokinin |
GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor. | |||
T34123 | Pranazepide | FR120480,FK 480,FR-120480 | cholecystokinin |
Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders and pancreatitis. | |||
T15382 | GI 181771 | cholecystokinin | |
GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity. | |||
T14932L1 | Ceruletide Ammonium Salt | Caerulein Ammonium Salt,Ceruletide Ammonium Salt(17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt | cholecystokinin |
Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is a potent cholecystokinin receptor agonist and a safe and effective cholecystokinin receptor agonist with direct spasmodic e... | |||
TP2030L1 | Gastrin I (human) acetate | Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate | cholecystokinin |
Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (CCK2) receptor. | |||
T9343 | N-Cbz-DL-tryptophan | cholecystokinin | |
N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8. | |||
T12404 | CCK-A receptor inhibitor 1 | cholecystokinin | |
T14932L | Ceruletide Ammonium acetate | FI-6934 Ammonium acetate,Caerulein Ammonium acetate,Ceruletide Ammonium acetate (17650-98-5 free base) | cholecystokinin |
Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist. Ceruletide Ammonium acetate is a safe and effective cholecystokinetic agent and small bowel and exocrine pancreatic stim... | |||
T26971 | Ceclazepide | ||
Ceclazepide is an antagonist of cholecystokinin receptor. | |||
T26483 | A-65186 | A65186 | |
A 65186 is a Type A Cholecystokinin (CCK) receptor antagonist. | |||
T24202 | Jmv 167 | Jmv-167,Jmv167 | |
Jmv 167 is an antagonist of the Cholecystokinin receptor. | |||
T23886 | Cholecystokinin (27-32)-amide | Cholecystokinin (27-32)-NH2 | |
Cholecystokinin (27-32)-amide is a CCK receptor antagonist. | |||
T29502 | A 70874 | A-70874,A70874 | |
A70874 has high selectivity and potency for cholecystokinin (CCK) a receptor. | |||
T28613 | RP73870 | RP 73870,RP-73870 | |
RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity. | |||
T25552 | Jmv 320 | Jmv-320,Jmv320 | |
Jmv 320 is a highly selective gastrin receptor and cholecystokinin receptor antagonist. It is a cyclic cholecystokinin-8 analog in which positions 28 and 31 have been replaced by Lys, with their side chains bridged by a ... | |||
T22895 | L-365260 | L-365,260 | Others |
cholecystokinin receptor 2 (CCK2) antagonist | |||
T13261 | CCK-B Receptor Antagonist 1 | Others | |
CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid. | |||
T24204 | Jmv 179 | Jmv-179,Jmv179 | |
Jmv 179 is an antagonist of the cholecystokinin receptor. | |||
T24293 | L 368935 | L-368935,L368,935,L-368,935,L 368,935,L368935 | |
L 368935 is an antagonist of the cholecystokinin receptor. | |||
T27664 | JNJ-17156516 | JNJ17156516,JNJ 17156516 | |
JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist. | |||
T28335 | PD 140376 | PD-140376,PD140376 | |
PD 140376 is a highly selective antagonist radioligand for the cholecystokinin(B)-gastrin receptor in guinea pig gastric mucosa & cerebral cortex in the peripheral and central nervous systems. | |||
T27669 | JNJ-26070109 | JNJ26070109 | |
JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat. | |||
T28331 | PD 136450 | Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189 | |
Cholecystokinin type B receptor antagonist PD-136,450 is a partial secretory agonist in the stomach and a full agonist in the pancreas of the rat. Gastrin (cholecystokinin type B (CCK-B)) receptor antagonists may help to... | |||
T68482 | CE-326597 | ||
CE-326597 is a potent and selective CCK1R agonist. The type 1 cholecystokinin receptor (CCK1R) has multiple physiologic roles relating to nutrient homeostasis,including mediation of postcibal satiety. The type 1 cholecy... | |||
T15101 | Devazepide | L-364,718,MK-329 | Others |
Devazepide is a competitive and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor (IC50s: 81 pM, 45 pM, and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respective... | |||
T17274 | YM022 | CCR | |
YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki v... | |||
T28612 | RP-72540 | RPR 102681,RPR-102681,RPR102681 | |
RP-72540 is a cholecystokinin B receptor antagonist. RP 72540 showed selectivity factors in express of 200 for CCKA versus CCKB receptors and also had high affinity for gastrin binding sites in the stomach. Administratio... | |||
T62039 | L-365260 hemihydrate | ||
L-365260 hemihydrate is a selective, orally active non-peptide gastrin and brain cholecystokinin receptor (CCK-B) antagonist, demonstrating competitive interaction with guinea pig stomach gastrin and brain CCK receptors ... | |||
T8761 | [Leu15]-Gastrin I human | Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2 | Others |
[Leu15]-Gastrin I human (Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2) encodes for the protein [Leu15]-Gastrin I in human. In human chromosome, the gene GAST is localized on... |
カタログ番号 | 製品名 | Species | Expression System |
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TMPH-03099 | Aminopeptidase N/CD13 Protein, Pig, Recombinant (His & Myc) | Sus scrofa (Pig) | E. coli |
Broad specificity aminopeptidase which plays a role in the final digestion of peptides generated from hydrolysis of proteins by gastric and pancreatic proteases. Also involved in the processing of various peptides includ... |